History of doping in sport / Charles E. Yesalis and Michael S. Bahrke
Determining the efficacy of performance-enhancing substances / Stan Reents
Anabolic-androgenic steroids / Michael S. Bahrke and Charles E. Yesalis
Beta-2 agonists / Gordon S. Lynch
Growth hormone : physiological effects of exogenous administration / William J. Kraemer, Bradley C. Nindl, and Martyn R. Rubin
Physiological effects of testosterone precursors / William J. Kraemer, Martyn R. Rubin, Duncan N. French, and Michael R. McGuigan
Human chorionic gonadotropin / R. Craig Kammerer.

Blood doping / Björn T. Ekblom
Erythropoietin / Björn T. Ekblom
Diuretics / Lawrence E. Armstrong
Narcotic analgesics and athletic performance / Dean F. Connors and John Sudkamp
Nonsteroidal anti-inflammatory drugs and corticosteroids / Louis C. Almekinders
Hypnotics, anxiolytics, and neuroleptics / Michael Bourin, Danièle Bentué-Ferrer, Hervé Allain, and Pierre Rochcongar
Beta-adrenergic antagonists / Kurt A. Mossberg and Claire Peel
Macronutrients and metabolic intermediates / Ellen Coleman and Suzanne Nelson Steen.

Creatine as an ergogenic supplement / J. David Branch and Melvin H. Williams
Sodium bicarbonate / Michael J. Webster
Herbals as ergogenic aids / Melvin H. Williams and J. David Branch
Alcohol usein sport and exercise / Robert D. Stainback and Rachelle Jansevics Cohen
Cannabis : clinical pharmacology and performance effects in humans / Stephen J. Heishman
Amphetamines / Steven B. Karch
Caffeine / Lawrence L. Spriet
Cocaine / Robert K. Conlee
Ephedrine as a ergogenic aid / Eric S. Rawson and Priscilla M. Clarkson.

Gamma-hydroxybutyric acid / Vincenzo R. Sanguineti and Marion Rudin Frank
Future and designer drugs : emerging science and technologies / Gary I. Wadler
Drug testing in sport and exercise / R. Craig Kammerer
Form over substances : the legal context of performance-enhancing substances / Charles E. Petit
Issues, concerns, and the future of performance-enhancing substances in sport and exercise / Michael S. Bahrke and Charles E. Yesalis.